Breakthrough therapies—
discovered faster than ever

Powered by an AI-native discovery engine and a relentless team, we turn complex chemistry into viable drug candidates across some of the toughest diseases—with speed and rigor.

We have built momentum from first experiments to a growing pipeline—and we’re only accelerating.

Many Inspithera molecules have
already advanced into R&D.
Watch their progress.

12 Development Candidates
01 Clinical Programs

CSM004

Mechanism: —

Indication: CNS

Granted

CSM045

Mechanism: —

Indication: Anti-Diabetes

Complete Filed

CSM050

Mechanism: —

Indication: Anti-Parkinson's

Complete Filed

CSM027

Mechanism: —

Indication: Hypertension

Provisional Filed

CSM046

Mechanism: —

Indication: Pain Management

Provisional Filed

CSM047

Mechanism: —

Indication: Pain Management

Provisional Filed

CSM048

Mechanism: —

Indication: Pain Management

Provisional Filed

CSM049

Mechanism: —

Indication: Appetite suppressant

Provisional Filed

CSM051

Mechanism: —

Indication: Anticonvulsant

Provisional Filed

CSM052

Mechanism: —

Indication: Pain Management

Provisional Filed

CSM053

Mechanism: —

Indication: CNS

Provisional Filed

CSM054

Mechanism: —

Indication: Antineoplastic

Provisional Filed

CSM055

Mechanism: —

Indication: Antiarrhythmic

Provisional Filed

CSM056

Mechanism: —

Indication: AntiCytomegalovirus

Provisional Filed

CSM057

Mechanism: —

Indication: Anticonvulsants

Provisional Filed

CSM058

Mechanism: —

Indication: Antineoplastic

Provisional Filed

CSM059

Mechanism: —

Indication: Antineoplastic

Provisional Filed

CSM060

Mechanism: —

Indication: Pain Management

Provisional Filed

CSM061

Mechanism: —

Indication: Hypertension

Provisional Filed

CSM062

Mechanism: —

Indication: Progesterone Antagonist

Provisional Filed

CSM063

Mechanism: —

Indication: CNS

Provisional Filed
Name
Mechanism
Indication
Discovery
Optimization
IND-Enabling
Phase 1
Phase 1b/2a
CSM004
—
CNS
 
 
 

CSM004 — Therapeutic Area: CNS. IP Status: Granted.

CSM045
—
Anti-Diabetes
 
 
 

CSM045 — Therapeutic Area: Anti-Diabetes. IP Status: Complete Filed.

CSM050
—
Anti-Parkinson's
 
 
 

CSM050 — Therapeutic Area: Anti-Parkinson’s. IP Status: Complete Filed.

CSM027
—
Hypertension
 
 
 

CSM027 — Therapeutic Area: Hypertension. IP Status: Provisional Filed.

CSM046
—
Pain Management
 
 
 

CSM046 — Therapeutic Area: Pain Management. IP Status: Provisional Filed.

CSM047
—
Pain Management
 
 
 

CSM047 — Therapeutic Area: Pain Management. IP Status: Provisional Filed.

CSM048
—
Pain Management
 
 
 

CSM048 — Therapeutic Area: Pain Management. IP Status: Provisional Filed.

CSM049
—
Appetite suppressant
 
 
 

CSM049 — Therapeutic Area: Appetite suppressant. IP Status: Provisional Filed.

CSM051
—
Anticonvulsant
 
 
 

CSM051 — Therapeutic Area: Anticonvulsant. IP Status: Provisional Filed.

CSM052
—
Pain Management
 
 
 

CSM052 — Therapeutic Area: Pain Management. IP Status: Provisional Filed.

CSM053
—
CNS
 
 
 

CSM053 — Therapeutic Area: CNS. IP Status: Provisional Filed.

CSM054
—
Antineoplastic
 
 
 

CSM054 — Therapeutic Area: Antineoplastic. IP Status: Provisional Filed.

CSM055
—
Antiarrhythmic
 
 
 

CSM055 — Therapeutic Area: Antiarrhythmic. IP Status: Provisional Filed.

CSM056
—
AntiCytomegalovirus
 
 
 

CSM056 — Therapeutic Area: AntiCytomegalovirus. IP Status: Provisional Filed.

CSM057
—
Anticonvulsants
 
 
 

CSM057 — Therapeutic Area: Anticonvulsants. IP Status: Provisional Filed.

CSM058
—
Antineoplastic
 
 
 

CSM058 — Therapeutic Area: Antineoplastic. IP Status: Provisional Filed.

CSM059
—
Antineoplastic
 
 
 

CSM059 — Therapeutic Area: Antineoplastic. IP Status: Provisional Filed.

CSM060
—
Pain Management
 
 
 

CSM060 — Therapeutic Area: Pain Management. IP Status: Provisional Filed.

CSM061
—
Hypertension
 
 
 

CSM061 — Therapeutic Area: Hypertension. IP Status: Provisional Filed.

CSM062
—
Progesterone Antagonist
 
 
 

CSM062 — Therapeutic Area: Progesterone Antagonist. IP Status: Provisional Filed.

CSM063
—
CNS
 
 
 

CSM063 — Therapeutic Area: CNS. IP Status: Provisional Filed.

  Development Candidate Declared

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Our focus today: therapeutics.
On the horizon: resilient agriculture, smarter nutrition, sustainable materials, and more.

By working together, we can rapidly expand the map of nature’s chemistry
and tackle pressing challenges across human and planetary health.
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